| Virtual screening-driven discovery of dual 5-HT6/5-HT2A receptor ligands with pro-cognitive properties J Staroń, R Kurczab, D Warszycki, G Satała, M Krawczyk, R Bugno, ... European Journal of Medicinal Chemistry 185, 111857, 2020 | 31 | 2020 |
| Search for a 5-CT alternative. In vitro and in vivo evaluation of novel pharmacological tools: 3-(1-alkyl-1 H-imidazol-5-yl)-1 H-indole-5-carboxamides, low-basicity 5-HT 7 … G Latacz, AS Hogendorf, A Hogendorf, A Lubelska, JM Wierońska, ... MedChemComm 9 (11), 1882-1890, 2018 | 30 | 2018 |
| Activation of the 5-HT7 receptor and MMP-9 signaling module in the hippocampal CA1 region is necessary for the development of depressive-like behavior M Bijata, E Bączyńska, FE Müller, K Bijata, J Masternak, A Krzystyniak, ... Cell Reports 38 (11), 2022 | 28 | 2022 |
| Design, synthesis, and biological evaluation of novel combretastatin A-4 thio derivatives as microtubule targeting agents T Stefański, R Mikstacka, R Kurczab, Z Dutkiewicz, M Kucińska, M Murias, ... European journal of medicinal chemistry 144, 797-816, 2018 | 26 | 2018 |
| 2-Aminoimidazole-based antagonists of the 5-HT6 receptor–A new concept in aminergic GPCR ligand design AS Hogendorf, A Hogendorf, R Kurczab, J Kalinowska-Tłuścik, P Popik, ... European Journal of Medicinal Chemistry 179, 1-15, 2019 | 25 | 2019 |
| Fluorinated indole-imidazole conjugates: Selective orally bioavailable 5-HT7 receptor low-basicity agonists, potential neuropathic painkillers AS Hogendorf, A Hogendorf, K Popiołek-Barczyk, A Ciechanowska, ... European Journal of Medicinal Chemistry 170, 261-275, 2019 | 25 | 2019 |
| 5-HT1A receptor ligands and their therapeutic applications: review of new patents J Staroń, R Bugno, AS Hogendorf, AJ Bojarski Expert Opinion on Therapeutic Patents 28 (9), 679-689, 2018 | 25 | 2018 |
| Regioselective hydroxylation of cholecalciferol, cholesterol and other sterol derivatives by steroid C25 dehydrogenase A Rugor, M Tataruch, J Staroń, A Dudzik, E Niedzialkowska, P Nowak, ... Applied microbiology and biotechnology 101, 1163-1174, 2017 | 21 | 2017 |
| Low-basicity 5-HT7 Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol AS Hogendorf, A Hogendorf, R Kurczab, G Satała, T Lenda, M Walczak, ... Scientific Reports 7 (1), 1444, 2017 | 19 | 2017 |
| Effects of ketamine optical isomers, psilocybin, psilocin and norpsilocin on time estimation and cognition in rats P Popik, A Hogendorf, R Bugno, SYS Khoo, P Zajdel, ... Psychopharmacology 239 (6), 1689-1703, 2022 | 16 | 2022 |
| Tuning the activity of known drugs via the introduction of halogen atoms, a case study of SERT ligands–Fluoxetine and fluvoxamine J Staroń, W Pietruś, R Bugno, R Kurczab, G Satała, D Warszycki, T Lenda, ... European Journal of Medicinal Chemistry 220, 113533, 2021 | 16 | 2021 |
| Distinct cognitive and discriminative stimulus effects of ketamine enantiomers in rats P Popik, SYS Khoo, A Kuziak, J Golebiowska, A Potasiewicz, ... Pharmacology Biochemistry and Behavior 197, 173011, 2020 | 11 | 2020 |
| Pyrano[2,3,4-cd]indole as a Scaffold for Selective Nonbasic 5-HT6R Ligands J Staroń, S Mordalski, D Warszycki, G Satała, A Hogendorf, AJ Bojarski ACS Medicinal Chemistry Letters 8 (4), 390-394, 2017 | 10 | 2017 |
| The effect of the intramolecular C–H⋯ O interactions on the conformational preferences of bis-arylsulfones–5-HT 6 receptor antagonists and beyond J Kalinowska-Tłuścik, J Staroń, A Krawczuk, S Mordalski, D Warszycki, ... RSC advances 8 (33), 18672-18681, 2018 | 8 | 2018 |
| How can fluorine directly and indirectly affect the hydrogen bonding in molecular systems?–A case study for monofluoroanilines W Pietruś, R Kurczab, R Kafel, E Machalska, J Kalinowska-Tłuścik, ... Spectrochimica Acta Part A: Molecular and Biomolecular Spectroscopy 252, 119536, 2021 | 6 | 2021 |
| Halogen bonding enhances activity in a series of dual 5-HT 6/D 2 ligands designed in a hybrid bioisostere generation/virtual screening protocol J Staroń, D Warszycki, R Kurczab, G Satała, R Bugno, A Hogendorf, ... RSC advances 6 (60), 54918-54925, 2016 | 6 | 2016 |
| Design and Synthesis of New Quinazolin-4-one Derivatives with Negative mGlu7 Receptor Modulation Activity and Antipsychotic-Like Properties K Kaczorowska, A Stankiewicz, R Bugno, MH Paluchowska, G Burnat, ... International Journal of Molecular Sciences 24 (3), 1981, 2023 | 5 | 2023 |
| Serotonin type 5A receptor antagonists inhibit D-lysergic acid diethylamide discriminatory cue in rats P Popik, M Krawczyk, A Kuziak, R Bugno, A Hogendorf, J Staroń, ... Journal of Psychopharmacology 33 (11), 1447-1455, 2019 | 5 | 2019 |
| N-Skatyltryptamines—Dual 5-HT6R/D2R Ligands with Antipsychotic and Procognitive Potential A Hogendorf, AS Hogendorf, R Kurczab, G Satała, B Szewczyk, P Cieślik, ... Molecules 26 (15), 4605, 2021 | 3 | 2021 |
| The effect of the intramolecular CH center dot center dot center dot O interactions on the conformational preferences of bis-arylsulfones-5-HT6 receptor antagonists and beyond J Kalinowska-Tluscik, J Staron, A Krawczuk, S Mordalski, D Warszycki, ... RSC ADVANCES 8 (33), 18672-18681, 2018 | 3 | 2018 |
Andrzej BojarskiMaj Institute of Pharmacology Polish Academy of SciencesVerified email at if-pan.krakow.pl
