| Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies M Bozdag, M Ferraroni, E Nuti, D Vullo, A Rossello, F Carta, A Scozzafava, ... Bioorganic & Medicinal Chemistry 22 (1), 334-340, 2014 | 112 | 2014 |
| 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors M Tanc, F Carta, M Bozdag, A Scozzafava, CT Supuran Bioorganic & medicinal chemistry 21 (15), 4502-4510, 2013 | 83 | 2013 |
| Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo [d] thiazole-5-and 6-sulfonamides M Abdoli, A Angeli, M Bozdag, F Carta, A Kakanejadifard, H Saeidian, ... Journal of Enzyme Inhibition and Medicinal Chemistry 32 (1), 1071-1078, 2017 | 59 | 2017 |
| Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups M Bozdag, M Ferraroni, F Carta, D Vullo, L Lucarini, E Orlandini, ... Journal of Medicinal Chemistry 57 (21), 9152-9167, 2014 | 59 | 2014 |
| Discovery of 4-hydroxy-3-(3-(phenylureido) benzenesulfonamides as SLC-0111 analogues for the treatment of hypoxic tumors overexpressing carbonic anhydrase IX M Bozdag, F Carta, M Ceruso, M Ferraroni, PC McDonald, S Dedhar, ... Journal of Medicinal Chemistry 61 (14), 6328-6338, 2018 | 57 | 2018 |
| A class of 4-sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects M Bozdag, M Pinard, F Carta, E Masini, A Scozzafava, R McKenna, ... Journal of Medicinal Chemistry 57 (22), 9673-9686, 2014 | 52 | 2014 |
| Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action M Bozdag, F Carta, D Vullo, A Akdemir, S Isik, C Lanzi, A Scozzafava, ... Bioorganic & Medicinal Chemistry 23 (10), 2368-2376, 2015 | 49 | 2015 |
| Selective inhibition of carbonic anhydrase IX over carbonic anhydrase XII in breast cancer cells using benzene sulfonamides: Disconnect between activity and growth inhibition MY Mboge, Z Chen, A Wolff, JV Mathias, C Tu, KD Brown, M Bozdag, ... PloS one 13 (11), e0207417, 2018 | 48 | 2018 |
| Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa D Vullo, S Del Prete, A Nocentini, SM Osman, Z AlOthman, C Capasso, ... Bioorganic & Medicinal Chemistry 25 (3), 1260-1265, 2017 | 48 | 2017 |
| Novel small molecule protein arginine deiminase 4 (PAD4) inhibitors M Bozdag, T Dreker, C Henry, P Tosco, M Vallaro, R Fruttero, ... Bioorganic & medicinal chemistry letters 23 (3), 715-719, 2013 | 42 | 2013 |
| Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity M Bozdag, AM Alafeefy, AM Altamimi, D Vullo, F Carta, CT Supuran Bioorganic & Medicinal Chemistry 25 (2), 677-683, 2017 | 41 | 2017 |
| Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis E Berrino, L Milazzo, L Micheli, D Vullo, A Angeli, M Bozdag, A Nocentini, ... Journal of Medicinal Chemistry 62 (15), 7233-7249, 2019 | 40 | 2019 |
| Carbonic anhydrase inhibitors based on sorafenib scaffold: design, synthesis, crystallographic investigation and effects on primary breast cancer cells M Bozdag, M Ferraroni, C Ward, F Carta, S Bua, A Angeli, SP Langdon, ... European Journal of Medicinal Chemistry 182, 111600, 2019 | 38 | 2019 |
| Azidothymidine “Clicked” into 1, 2, 3-triazoles: first report on carbonic anhydrase–telomerase dual-hybrid inhibitors E Berrino, A Angeli, DD Zhdanov, AP Kiryukhina, A Milaneschi, A De Luca, ... Journal of medicinal chemistry 63 (13), 7392-7409, 2020 | 32 | 2020 |
| A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells MY Mboge, Z Chen, D Khokhar, A Wolff, L Ai, CD Heldermon, M Bozdag, ... Biochemical Journal 476 (10), 1497-1513, 2019 | 32 | 2019 |
| Pain relieving effect of-NSAIDs-CAIs hybrid molecules: Systemic and intra-articular treatments against rheumatoid arthritis L Micheli, M Bozdag, O Akgul, F Carta, C Guccione, MC Bergonzi, ... International journal of molecular sciences 20 (8), 1923, 2019 | 32 | 2019 |
| Synthesis of a novel affinity gel for the purification of carbonic anhydrases M Bozdag, S Isik, S Beyaztas, O Arslan, CT Supuran Journal of enzyme inhibition and medicinal chemistry 30 (2), 240-244, 2015 | 32 | 2015 |
| Mycobacterium tuberculosisβ-Carbonic Anhydrases: Novel Targets for Developing Antituberculosis Drugs A Aspatwar, V Kairys, S Rala, M Parikka, M Bozdag, F Carta, CT Supuran, ... International Journal of Molecular Sciences 20 (20), 5153, 2019 | 30 | 2019 |
| “A sweet combination”: developing saccharin and acesulfame K structures for selectively targeting the tumor-associated carbonic anhydrases IX and XII S Bua, C Lomelino, AB Murray, SM Osman, ZA ALOthman, M Bozdag, ... Journal of Medicinal Chemistry 63 (1), 321-333, 2019 | 28 | 2019 |
| Novel 6-and 7-substituted coumarins with inhibitory action against lipoxygenase and tumor-associated carbonic anhydrase IX A Peperidou, S Bua, M Bozdag, D Hadjipavlou-Litina, CT Supuran Molecules 23 (1), 153, 2018 | 28 | 2018 |
Fabrizio CartaUniversita' di Firenze-Dept. NeurofarbaVerified email at unifi.it
