Giovanni Piersanti
Giovanni Piersanti
Professor of Organic Chemistry, UniveritÓ di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari
Verified email at uniurb.it - Homepage
TitleCited byYear
Cyclohexylcarbamic acid 3 ‘-or 4 ‘-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: Synthesis, quantitative structure− activity relationships, andá…
M Mor, S Rivara, A Lodola, PV Plazzi, G Tarzia, A Duranti, A Tontini, ...
Journal of medicinal chemistry 47 (21), 4998-5008, 2004
2752004
Design, synthesis, and structure− activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors
G Tarzia, A Duranti, A Tontini, G Piersanti, M Mor, S Rivara, PV Plazzi, ...
Journal of medicinal chemistry 46 (12), 2352-2360, 2003
1832003
2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacologicalá…
P Minetti, MO Tinti, P Carminati, M Castorina, MA Di Cesare, S Di Serio, ...
Journal of medicinal chemistry 48 (22), 6887-6896, 2005
882005
Synthesis and quantitative structure− activity relationship of fatty acid amide hydrolase inhibitors: modulation at the N-portion of biphenyl-3-yl alkylcarbamates
M Mor, A Lodola, S Rivara, F Vacondio, A Duranti, A Tontini, S Sanchini, ...
Journal of medicinal chemistry 51 (12), 3487-3498, 2008
682008
Synthesis and structure–activity relationships of FAAH inhibitors: cyclohexylcarbamic acid biphenyl esters with chemical modulation at the proximal phenyl ring
G Tarzia, A Duranti, G Gatti, G Piersanti, A Tontini, S Rivara, A Lodola, ...
ChemMedChem: Chemistry Enabling Drug Discovery 1 (1), 130-139, 2006
662006
Enantioselective Total Synthesis of (−)‐Acylfulvene and (−)‐Irofulven
M Movassaghi, G Piizzi, DS Siegel, G Piersanti
Angewandte Chemie International Edition 45 (35), 5859-5863, 2006
652006
Switchable Reactivity of Acylated α, β-Dehydroamino Ester in the Friedel− Crafts Alkylation of Indoles by Changing the Lewis Acid
E Angelini, C Balsamini, F Bartoccini, S Lucarini, G Piersanti
The Journal of organic chemistry 73 (14), 5654-5657, 2008
622008
Enantioselective Total Synthesis of (−)-Acylfulvene and (−)-Irofulven
DS Siegel, G Piizzi, G Piersanti, M Movassaghi
The Journal of organic chemistry 74 (24), 9292-9304, 2009
512009
Quantifying amino acid conformational preferences and side-chain–side-chain interactions in β-hairpins
ST Phillips, G Piersanti, PA Bartlett
Proceedings of the National Academy of Sciences 102 (39), 13737-13742, 2005
512005
Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2A Antagonists/MAO-B Inhibitors
S Rivara, G Piersanti, F Bartoccini, G Diamantini, D Pala, T Riccioni, ...
Journal of medicinal chemistry 56 (3), 1247-1261, 2013
432013
A Trans-Stereoselective Synthesis of 3-Halo-4-alkyl (aryl)-NH-azetidin-2-ones
E Bandini, G Favi, G Martelli, M Panunzio, G Piersanti
Organic letters 2 (8), 1077-1079, 2000
422000
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (▒)-Esermethole
S Lucarini, F Bartoccini, F Battistoni, G Diamantini, G Piersanti, M Righi, ...
Organic letters 12 (17), 3844-3847, 2010
402010
Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles
M Righi, F Topi, S Bartolucci, A Bedini, G Piersanti, G Spadoni
The Journal of organic chemistry 77 (14), 6351-6357, 2012
392012
Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity
V Lucini, M Pannacci, F Scaglione, F Fraschini, S Rivara, M Mor, F Bordi, ...
Journal of medicinal chemistry 47 (17), 4202-4212, 2004
372004
New branched macrocyclic ligand and its side-arm, two urea-based receptors for anions: synthesis, binding studies and crystal structure
M Formica, V Fusi, E Macedi, P Paoli, G Piersanti, P Rossi, G Zappia, ...
New Journal of Chemistry 32 (7), 1204-1214, 2008
342008
Synthesis of (−)-Epi-Indolactam V by an Intramolecular Buchwald–Hartwig C–N Coupling Cyclization Reaction
M Mari, F Bartoccini, G Piersanti
The Journal of organic chemistry 78 (15), 7727-7734, 2013
302013
Iridium-catalyzed direct synthesis of tryptamine derivatives from indoles: exploiting N-protected β-amino alcohols as alkylating agents
S Bartolucci, M Mari, A Bedini, G Piersanti, G Spadoni
The Journal of organic chemistry 80 (6), 3217-3222, 2015
272015
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation
S Bartolucci, F Bartoccini, M Righi, G Piersanti
Organic letters 14 (2), 600-603, 2012
272012
New coumarin-urea based receptor for anions: A selective off–on fluorescence response to fluoride
G Ambrosi, M Formica, V Fusi, L Giorgi, E Macedi, G Piersanti, M Retini, ...
Tetrahedron 68 (19), 3768-3775, 2012
262012
Stereochemical Aspects of a Two‐Step Staudinger Reaction− Asymmetric Synthesis of Chiral Azetidine‐2‐ones
A Bongini, M Panunzio, G Piersanti, E Bandini, G Martelli, G Spunta, ...
European Journal of Organic Chemistry 2000 (13), 2379-2390, 2000
262000
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