Design, synthesis and characterization of novel 1, 2-benzisothiazol-3 (2H)-one and 1, 3, 4-oxadiazole hybrid derivatives: potent inhibitors of Dengue and West Nile virus NS2B … H Lai, D Dou, S Aravapalli, T Teramoto, GH Lushington, TM Mwania, ... Bioorganic & medicinal chemistry 21 (1), 102-113, 2013 | 68 | 2013 |
Design, synthesis, and evaluation of inhibitors of Norwalk virus 3C protease KC Tiew, G He, S Aravapalli, SR Mandadapu, MR Gunnam, KR Alliston, ... Bioorganic & medicinal chemistry letters 21 (18), 5315-5319, 2011 | 67 | 2011 |
Macrocyclic inhibitors of 3C and 3C-like proteases of picornavirus, norovirus, and coronavirus SR Mandadapu, PM Weerawarna, AM Prior, RAZ Uy, S Aravapalli, ... Bioorganic & medicinal chemistry letters 23 (13), 3709-3712, 2013 | 59 | 2013 |
Inhibitors of Dengue virus and West Nile virus proteases based on the aminobenzamide scaffold S Aravapalli, H Lai, T Teramoto, KR Alliston, GH Lushington, EL Ferguson, ... Bioorganic & medicinal chemistry 20 (13), 4140-4148, 2012 | 57 | 2012 |
Inhibition of noroviruses by piperazine derivatives D Dou, G He, SR Mandadapu, S Aravapalli, Y Kim, KO Chang, ... Bioorganic & medicinal chemistry letters 22 (1), 377-379, 2012 | 56 | 2012 |
Antifungal activity of a series of 1, 2-benzisothiazol-3 (2H)-one derivatives D Dou, D Alex, B Du, KC Tiew, S Aravapalli, SR Mandadapu, ... Bioorganic & medicinal chemistry 19 (19), 5782-5787, 2011 | 41 | 2011 |
Potent inhibition of Norwalk virus by cyclic sulfamide derivatives D Dou, KC Tiew, G He, SR Mandadapu, S Aravapalli, KR Alliston, Y Kim, ... Bioorganic & medicinal chemistry 19 (20), 5975-5983, 2011 | 35 | 2011 |
Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening AJA Woolford, JE Pero, S Aravapalli, V Berdini, JE Coyle, PJ Day, ... Journal of Medicinal Chemistry 59 (11), 5356-5367, 2016 | 23 | 2016 |
Effects of chamber pressure and partial pressure of water vapor on secondary drying in lyophilization JA Searles, S Aravapalli, C Hodge AAPS PharmSciTech 18 (7), 2808-2813, 2017 | 14 | 2017 |
Discovery of a novel binder of Lp-PLA2 and subsequent optimization through rational target design J Pero, S Aravapalli, V Berdini, J Coyle, P Day, A Dodson, P Grondin, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 252, 2016 | | 2016 |
Discovery and optimization of novel chemotype LpPLA2 inhibitors featuring a unique binding mode P Li, S Aravapalli, A Dodson, B McCleland, E Manas, J Marino, C Neipp, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 252, 2016 | | 2016 |