| Discovery of Chemoselective and Biocompatible Reactions Using a High‐Throughput Immunoassay Screening S Kolodych, E Rasolofonjatovo, M Chaumontet, MC Nevers, C Créminon, ... Angewandte Chemie International Edition 52 (46), 12056-12060, 2013 | 138 | 2013 |
| Ultrafast Click Chemistry with Fluorosydnones H Liu, D Audisio, L Plougastel, E Decuypere, DA Buisson, O Koniev, ... Angewandte Chemie International Edition 55 (39), 12073-12077, 2016 | 116 | 2016 |
| Iridium-Catalyzed Cycloaddition of Azides and 1-Bromoalkynes at Room Temperature E Rasolofonjatovo, S Theeramunkong, A Bouriaud, S Kolodych, ... Organic letters 15 (18), 4698-4701, 2013 | 111 | 2013 |
| Antibody–Oligonucleotide Conjugates as Therapeutic, Imaging, and Detection Agents I Dovgan, O Koniev, S Kolodych, A Wagner Bioconjugate chemistry 30 (10), 2483-2501, 2019 | 110 | 2019 |
| Targeting the tumour microenvironment with an enzyme-responsive drug delivery system for the efficient therapy of breast and pancreatic cancers B Renoux, F Raes, T Legigan, E Péraudeau, B Eddhif, P Poinot, ... Chemical Science 8 (5), 3427-3433, 2017 | 110 | 2017 |
| Bioorthogonal Click and Release Reaction of Iminosydnones with Cycloalkynes S Bernard, D Audisio, M Riomet, S Bregant, A Sallustrau, L Plougastel, ... Angewandte Chemie International Edition 56 (49), 15612-15616, 2017 | 100 | 2017 |
| 4-Halogeno-sydnones for fast strain promoted cycloaddition with bicyclo-[6.1. 0]-nonyne L Plougastel, O Koniev, S Specklin, E Decuypere, C Créminon, ... Chemical Communications 50 (66), 9376-9378, 2014 | 93 | 2014 |
| CBTF: New amine-to-thiol coupling reagent for preparation of antibody conjugates with increased plasma stability S Kolodych, O Koniev, Z Baatarkhuu, JY Bonnefoy, F Debaene, ... Bioconjugate chemistry 26 (2), 197-200, 2015 | 78 | 2015 |
| Development and evaluation of β-galactosidase-sensitive antibody-drug conjugates S Kolodych, C Michel, S Delacroix, O Koniev, A Ehkirch, J Eberova, ... European Journal of Medicinal Chemistry, 2017 | 67 | 2017 |
| Copper (I)-Catalyzed Cycloaddition of 4-Bromosydnones and Alkynes for the Regioselective Synthesis of 1, 4, 5-Trisubstituted Pyrazoles E Decuypere, S Specklin, S Gabillet, D Audisio, H Liu, L Plougastel, ... Organic letters 17 (2), 362-365, 2015 | 60 | 2015 |
| Palladium‐Catalyzed Chemoselective and Biocompatible Functionalization of Cysteine‐Containing Molecules at Room Temperature RAA Al‐Shuaeeb, S Kolodych, O Koniev, S Delacroix, S Erb, S Nicolaÿ, ... Chemistry-A European Journal 22 (32), 11365-11370, 2016 | 55 | 2016 |
| 2-(Maleimidomethyl)-1, 3-Dioxanes (MD): a Serum-Stable Self-hydrolysable Hydrophilic Alternative to Classical Maleimide Conjugation I Dovgan, S Kolodych, O Koniev, A Wagner Scientific Reports 6, 2016 | 54 | 2016 |
| Acyl Fluorides: Fast, Efficient, and Versatile Lysine-Based Protein Conjugation via Plug-and-Play Strategy I Dovgan, S Ursuegui, S Erb, C Michel, S Kolodych, S Cianférani, ... Bioconjugate Chemistry 28 (5), 1452-1457, 2017 | 51 | 2017 |
| Reaction Discovery by Using a Sandwich Immunoassay J Quinton, S Kolodych, M Chaumonet, V Bevilacqua, MC Nevers, ... Angewandte Chemie International Edition 51 (25), 6144-6148, 2012 | 44 | 2012 |
| Reduction–rebridging strategy for the preparation of ADPN-based antibody–drug conjugates O Koniev, I Dovgan, B Renoux, A Ehkirch, J Eberova, S Cianférani, ... MedChemComm 9 (5), 827-830, 2018 | 37 | 2018 |
| Design and Synthesis of Iminosydnones for Fast Click and Release Reactions with Cycloalkynes M Riomet, E Decuypere, K Porte, S Bernard, L Plougastel, S Kolodych, ... Chemistry–A European Journal 24 (34), 8535-8541, 2018 | 35 | 2018 |
| On the use of DNA as a linker in antibody-drug conjugates: synthesis, stability and in vitro potency I Dovgan, A Ehkirch, V Lehot, I Kuhn, O Koniev, S Kolodych, A Hentz, ... Scientific Reports 10 (1), 1-9, 2020 | 24 | 2020 |
| Automated linkage of proteins and payloads producing monodisperse conjugates I Dovgan, A Hentz, O Koniev, A Ehkirch, S Hessmann, S Ursuegui, ... Chemical Science 11 (5), 1210-1215, 2020 | 20 | 2020 |
| MAPN: First-in-class reagent for kinetically resolved thiol-to-thiol conjugation O Koniev, S Kolodych, Z Baatarkhuu, J Stojko, J Eberova, JY Bonnefoy, ... Bioconjugate Chemistry 26 (9), 1863-1867, 2015 | 18 | 2015 |
| An Efficient Synthesis of Fused 3-Formylpyridines and 5-Formylpyrimidines AP Mityuk, SE Kolodych, SA Mytnyk, YV Dmytriv, DM Volochnyuk, ... Synthesis 2010 (16), 2767-2770, 2010 | 14 | 2010 |
Oleksandr KonievSyndiviaVerified email at syndivia.com
