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Adel S. El-Azab
Adel S. El-Azab
Other namesAdel S. ElAzab,, Adel S. Al-Azab
Unknown affiliation
Verified email at Ksu.edu.sa
Title
Cited by
Cited by
Year
Design, synthesis and biological evaluation of novel quinazoline derivatives as potential antitumor agents: molecular docking study
AS El-Azab, MA Al-Omar, AM Alaa, NI Abdel-Aziz, AA Magda, AM Aleisa, ...
European journal of medicinal chemistry 45 (9), 4188-4198, 2010
2882010
Substituted quinazolines, part 3. Synthesis, in vitro antitumor activity and molecular modeling study of certain 2-thieno-4 (3H)-quinazolinone analogs
AM Al-Obaid, SG Abdel-Hamide, HA El-Kashef, AM Alaa, AS El-Azab, ...
European journal of medicinal chemistry 44 (6), 2379-2391, 2009
2162009
Design, synthesis, and biological evaluation of substituted hydrazone and pyrazole derivatives as selective COX-2 inhibitors: Molecular docking study
AA Magda, NI Abdel-Aziz, AM Alaa, AS El-Azab, YA Asiri, KEH ElTahir
Bioorganic & medicinal chemistry 19 (11), 3416-3424, 2011
1812011
Synthesis, biological evaluation and molecular modeling study of pyrazole and pyrazoline derivatives as selective COX-2 inhibitors and anti-inflammatory agents. Part 2
AA Magda, NI Abdel-Aziz, AM Alaa, AS El-Azab, KEH ElTahir
Bioorganic & medicinal chemistry 20 (10), 3306-3316, 2012
1712012
Non-classical antifolates. Part 2: synthesis, biological evaluation, and molecular modeling study of some new 2, 6-substituted-quinazolin-4-ones
FAM Al-Omary, LA Abou-Zeid, MN Nagi, ESE Habib, AM Alaa, AS El-Azab, ...
Bioorganic & medicinal chemistry 18 (8), 2849-2863, 2010
1632010
Structure-based design of phthalimide derivatives as potential cyclooxygenase-2 (COX-2) inhibitors: anti-inflammatory and analgesic activities
AM Alanazi, AS El-Azab, IA Al-Suwaidan, KEH ElTahir, YA Asiri, ...
European journal of medicinal chemistry 92, 115-123, 2015
1302015
Synthesis and anticonvulsant evaluation of some new 2, 3, 8-trisubstituted-4 (3H)-quinazoline derivatives
AS El-Azab, KEH ElTahir
Bioorganic & medicinal chemistry letters 22 (1), 327-333, 2012
1042012
Design and synthesis of novel 7-aminoquinazoline derivatives: Antitumor and anticonvulsant activities
AS El-Azab, KEH ElTahir
Bioorganic & medicinal chemistry letters 22 (5), 1879-1885, 2012
1012012
Synthesis, anti-inflammatory, analgesic, COX-1/2 inhibitory activities and molecular docking studies of substituted 2-mercapto-4 (3H)-quinazolinones
AM Alaa, LA Abou-Zeid, KEH ElTahir, RR Ayyad, AA Magda, AS El-Azab
European Journal of Medicinal Chemistry 121, 410-421, 2016
1002016
Synthesis and antitumor evaluation of trimethoxyanilides based on 4 (3H)-quinazolinone scaffolds
MA Mohamed, RR Ayyad, TZ Shawer, AM Alaa, AS El-Azab
European journal of medicinal chemistry 112, 106-113, 2016
902016
Design, synthesis of 2, 3-disubstitued 4 (3H)-quinazolinone derivatives as anti-inflammatory and analgesic agents: COX-1/2 inhibitory activities and molecular docking studies
AM Alaa, LA Abou-Zeid, KEH ElTahir, MA Mohamed, MAA El-Enin, ...
Bioorganic & Medicinal Chemistry 24 (16), 3818-3828, 2016
772016
Synthesis, antitumor activity and molecular docking study of some novel 3-benzyl-4 (3H) quinazolinone analogues
IA Al-Suwaidan, AAM Abdel-Aziz, TZ Shawer, RR Ayyad, AM Alanazi, ...
Journal of enzyme inhibition and medicinal chemistry 31 (1), 78-89, 2016
762016
Synthesis and biological evaluation of some novel cyclic-imides as hypoglycaemic, anti-hyperlipidemic agents
AM Alaa, AS El-Azab, SM Attia, AM Al-Obaid, MA Al-Omar, HI El-Subbagh
European journal of medicinal chemistry 46 (9), 4324-4329, 2011
732011
Design, synthesis and biological evaluation of some novel substituted quinazolines as antitumor agents
AM Alanazi, AM Alaa, IA Al-Suwaidan, SG Abdel-Hamide, TZ Shawer, ...
European journal of medicinal chemistry 79, 446-454, 2014
722014
Design, synthesis and biological evaluation of 2-mercapto-3-phenethylquinazoline bearing anilide fragments as potential antitumor agents: molecular docking study
IA Al-Suwaidan, AM Alanazi, AM Alaa, MA Mohamed, AS El-Azab
Bioorganic & medicinal chemistry letters 23 (13), 3935-3941, 2013
712013
Synthesis and anti-inflammatory activity of sulfonamides and carboxylates incorporating trimellitimides: dual cyclooxygenase/carbonic anhydrase inhibitory actions
AM Alaa, A Angeli, AS El-Azab, MEA Hammouda, MA El-Sherbeny, ...
Bioorganic chemistry 84, 260-268, 2019
652019
Acacia Senegal gum exudate offers protection against cyclophosphamide-induced urinary bladder cytotoxicity
AA Al-Yahya, AA Al-Majed, AM Gado, MH Daba, OA Al-Shabanah, ...
Oxidative medicine and cellular longevity 2, 207-213, 2009
652009
Synthesis and potential antitumor activity of 7-(4-substituted piperazin-1-yl)-4-oxoquinolines based on ciprofloxacin and norfloxacin scaffolds: in silico studies
AAM Abdel-Aziz, AS El-Azab, AM Alanazi, YA Asiri, IA Al-Suwaidan, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (5), 796-809, 2016
642016
Molecular design, synthesis and biological evaluation of cyclic imides bearing benzenesulfonamide fragment as potential COX-2 inhibitors. Part 2
IA Al-Suwaidan, AM Alanazi, AS El-Azab, AM Al-Obaid, KEH ElTahir, ...
Bioorganic & medicinal chemistry letters 23 (9), 2601-2605, 2013
642013
Synthesis, anti-inflammatory, analgesic and COX-1/2 inhibition activities of anilides based on 5, 5-diphenylimidazolidine-2, 4-dione scaffold: molecular docking studies
AM Alaa, AS El-Azab, LA Abou-Zeid, KEH ElTahir, NI Abdel-Aziz, ...
European journal of medicinal chemistry 115, 121-131, 2016
622016
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