| Macrocyclization of Peptide Side Chains by the Ugi Reaction: Achieving Peptide Folding and Exocyclic N-Functionalization in One Shot AV Vasco, CS Pérez, FE Morales, HE Garay, D Vasilev, JA Gavin, ... The Journal of Organic Chemistry 80 (13), 6697-6707, 2015 | 64 | 2015 |
| A Multicomponent Conjugation Strategy to Unique N‐Steroidal Peptides: First Evidence of the Steroidal Nucleus as a β‐Turn Inducer in Acyclic Peptides DG Rivera, AV Vasco, R Echemendía, O Concepción, CS Pérez, JA Gavín, ... Chemistry–A European Journal 20 (41), 13150-13161, 2014 | 57 | 2014 |
| Multicomponent polysaccharide–protein bioconjugation in the development of antibacterial glycoconjugate vaccine candidates Y Méndez, J Chang, AR Humpierre, A Zanuy, R Garrido, AV Vasco, ... Chemical science 9 (9), 2581-2588, 2018 | 52 | 2018 |
| A multicomponent stapling approach to exocyclic functionalized helical peptides: adding lipids, sugars, PEGs, labels, and handles to the lactam bridge AV Vasco, Y Méndez, A Porzel, J Balbach, LA Wessjohann, DG Rivera Bioconjugate Chemistry 30 (1), 253-259, 2018 | 48 | 2018 |
| Discovery of potent and selective inhibitors of the Escherichia coli M1-aminopeptidase via multicomponent solid-phase synthesis of tetrazole-peptidomimetics Y Méndez, G De Armas, I Pérez, T Rojas, ME Valdés-Tresanco, ... European Journal of Medicinal Chemistry 163, 481-499, 2019 | 38 | 2019 |
| Expanding the scope of Ugi multicomponent bioconjugation to produce pneumococcal multivalent glycoconjugates as vaccine candidates AR Humpierre, A Zanuy, M Saenz, R Garrido, AV Vasco, R Pérez-Nicado, ... Bioconjugate Chemistry 31 (9), 2231-2240, 2020 | 19 | 2020 |
| Stabilization of Cyclic β-Hairpins by Ugi-Reaction-Derived N-Alkylated Peptides: The Quest for Functionalized β-Turns MG Ricardo, AV Vasco, DG Rivera, LA Wessjohann Organic letters 21 (18), 7307-7310, 2019 | 19 | 2019 |
| On-resin multicomponent protocols for biopolymer assembly and derivatization DG Rivera, MG Ricardo, AV Vasco, LA Wessjohann, EV Van der Eycken Nature Protocols 16 (2), 561-578, 2021 | 16 | 2021 |
| Synthesis of lactam-bridged and lipidated cyclo-peptides as promising anti-phytopathogenic agents AV Vasco, M Brode, Y Méndez, O Valdés, DG Rivera, LA Wessjohann Molecules 25 (4), 811, 2020 | 14 | 2020 |
| Isonitriles: versatile handles for the bioorthogonal functionalization of proteins Y Méndez, AV Vasco, AR Humpierre, B Westermann ACS omega 5 (40), 25505-25510, 2020 | 8 | 2020 |
| Iridoids and volatile pheromones of Tapinoma darioi ants: chemical differences to the closely related species Tapinoma magnum D D’Eustacchio, M Centorame, A Fanfani, G Senczuk, ... Chemoecology 29, 51-60, 2019 | 8 | 2019 |
| Total synthesis of cordyheptapeptide A AR Puentes, RAW Neves Filho, DG Rivera, LA Wessjohann Synlett 28 (15), 1971-1974, 2017 | 7 | 2017 |
| ERp57 chaperon protein protects neuronal cells from Aβ‐induced toxicity D Di Risola, D Ricci, I Marrocco, F Giamogante, M Grieco, A Francioso, ... Journal of Neurochemistry 162 (4), 322-336, 2022 | 6 | 2022 |
| Insights into the secondary structures of lactam N-substituted stapled peptides AV Vasco, CG Moya, S Gröger, W Brandt, J Balbach, CS Pérez, ... Organic & Biomolecular Chemistry 18 (20), 3838-3842, 2020 | 6 | 2020 |
| Merging the Isonitrile‐Tetrazine (4+ 1) Cycloaddition and the Ugi Four‐Component Reaction into a Single Multicomponent Process Y Méndez, AV Vasco, G Ivey, AL Dias, P Gierth, BB Sousa, CD Navo, ... Angewandte Chemie International Edition 62 (44), e202311186, 2023 | 1 | 2023 |
| Multicomponent Functionalization of the Octreotide Peptide Macrocyclic Scaffold AV Vasco, LG Ceballos, LA Wessjohann, DG Rivera European Journal of Organic Chemistry 2022 (39), e202200687, 2022 | 1 | 2022 |
| Quantitative NMR for the structural analysis of novel bivalent glycoconjugates as vaccine candidates AR Humpierre, A Zanuy, M Saenz, AV Vasco, Y Méndez, B Westermann, ... Journal of Pharmaceutical and Biomedical Analysis 214, 114721, 2022 | 1 | 2022 |
| Ligation, Macrocyclization, and Simultaneous Functionalization of Peptides by Multicomponent Reactions (MCR) AV Vasco, MG Ricardo, DG Rivera, LA Wessjohann Peptide Macrocycles: Methods and Protocols, 143-157, 2022 | 1 | 2022 |
| Frontispiece: A Multicomponent Conjugation Strategy to Unique N‐Steroidal Peptides: First Evidence of the Steroidal Nucleus as a β‐Turn Inducer in Acyclic Peptides DG Rivera, AV Vasco, R Echemendía, O Concepción, CS Pérez, JA Gavín, ... Chemistry–A European Journal 20 (41), 2014 | 1 | 2014 |
| Cathepsin B Processing Is Required for the In Vivo Efficacy of Albumin–Drug Conjugates B Bernardim, J Conde, T Hakala, JB Becher, M Canzano, AV Vasco, ... Bioconjugate Chemistry, 2024 | | 2024 |
