Paul Glossop
Paul Glossop
Sandexis
Verified email at sandexis.co.uk
TitleCited byYear
Inhalation by design: novel ultra-long-acting β2-adrenoreceptor agonists for inhaled once-daily treatment of asthma and chronic obstructive pulmonary disease that utilize a …
PA Glossop, CAL Lane, DA Price, ME Bunnage, RA Lewthwaite, K James, ...
Journal of medicinal chemistry 53 (18), 6640-6652, 2010
652010
Stereoselective synthesis of pyrrolidines: catalytic oxidative cyclizations mediated by osmium
TJ Donohoe, GH Churchill, PA Glossop
Angewandte Chemie 118 (47), 8193-8196, 2006
522006
The discovery of long acting β< sub> 2</sub>-adrenoreceptor agonists
AD Brown, ME Bunnage, PA Glossop, K James, R Jones, CAL Lane, ...
Bioorganic & medicinal chemistry letters 17 (14), 4012-4015, 2007
492007
Pyridine‐N‐Oxide as a Mild Reoxidant Which Transforms Osmium‐Catalyzed Oxidative Cyclization
TJ Donohoe, PJ Lindsay‐Scott, PA Glossop, IA Nash, JS Parker
Angewandte Chemie 120 (15), 2914-2917, 2008
372008
Inhibition of TRPM8 channels reduces pain in the cold pressor test in humans
WJ Winchester, K Gore, S Glatt, W Petit, JC Gardiner, K Conlon, ...
Journal of Pharmacology and Experimental Therapeutics 351 (2), 259-269, 2014
352014
The discovery of adamantyl-derived, inhaled, long acting β< sub> 2</sub>-adrenoreceptor agonists
AD Brown, ME Bunnage, PA Glossop, K James, R Jones, CAL Lane, ...
Bioorganic & medicinal chemistry letters 18 (4), 1280-1283, 2008
352008
The discovery of indole-derived long acting β< sub> 2</sub>-adrenoceptor agonists for the treatment of asthma and COPD
AD Brown, ME Bunnage, PA Glossop, M Holbrook, RD Jones, CAL Lane, ...
Bioorganic & medicinal chemistry letters 17 (22), 6188-6191, 2007
282007
Inhalation by design: novel tertiary amine muscarinic m3 receptor antagonists with slow off-rate binding kinetics for inhaled once-daily treatment of chronic obstructive …
PA Glossop, CAL Watson, DA Price, ME Bunnage, DS Middleton, A Wood, ...
Journal of medicinal chemistry 54 (19), 6888-6904, 2011
252011
Progress in the Development of Inhaled, Long-Acting b2-Adrenoceptor Agonists
PA Glossop, DA Price
Annual Reports in Medicinal Chemistry 41, 237, 2006
212006
Identification of Type‐II Inhibitors Using Kinase Structures
F Lovering, J McDonald, GA Whitlock, PA Glossop, C Phillips, A Bent, ...
Chemical Biology & Drug Design 80 (5), 657-664, 2012
182012
COMPOUNDS HAVING BETA-AGONIST ACTIVITY
A BROWN, M BUNNAGE, K BUTCHER, P GLOSSOP, K JAMES, C LANE, ...
WO Patent 2,005,092,841, 2005
18*2005
Osmium‐Mediated Oxidative Cyclizations: A Study into the Range of Initiators That Facilitate Cyclization
TJ Donohoe, PJ Lindsay‐Scott, GH Churchill, MJ Connolly, S Butterworth, ...
Chemistry–An Asian Journal 4 (8), 1237-1247, 2009
152009
Studies on DMDO-mediated benzylidene acetal oxidation
DK Mycock, AE Sherlock, PA Glossop, CJ Hayes
Tetrahedron Letters 49 (45), 6390-6392, 2008
152008
Designing rapid onset selective serotonin re-uptake inhibitors. Part 1: Structure–activity relationships of substituted (1< i> S</i>, 4< i> S</i>)-4-(3, 4-dichlorophenyl)-< i …
DS Middleton, M Andrews, P Glossop, G Gymer, A Jessiman, PS Johnson, ...
Bioorganic & medicinal chemistry letters 16 (5), 1434-1439, 2006
142006
Development of a Scaleable Synthesis of a Geminal Dimethyl Tertiary Amine as an Inhaled Muscarinic Antagonist for the Treatment of COPD
BR Dillon, DF Roberts, DA Entwistle, PA Glossop, CJ Knight, DA Laity, ...
Organic Process Research & Development 16 (2), 195-203, 2012
132012
NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS
SP Bailey, CG Barber, PA Glossop, DS Middleton
EP Patent 1,651,609, 2006
132006
Design and synthesis of long acting inhaled corticosteroids for the treatment of asthma
DS Millan, SA Ballard, S Chunn, JA Dybowski, CK Fulton, PA Glossop, ...
Bioorganic & medicinal chemistry letters 21 (19), 5826-5830, 2011
122011
Compounds useful for the treatment of diseases
ME Bunnage, PA Glossop, CAL Lane, RA Lewthwaite
US Patent 7,268,147, 2007
112007
Indole derivatives useful for the treatment of diseases
AD Brown, JS Bryans, ME Bunnage, PA Glossop, CAL Lane, ...
US Patent 7,138,527, 2006
112006
NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS
S BAILEY, C BARBER, P GLOSSOP, D MIDDLETON
WO Patent 2,005,009,966, 2005
102005
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