Matthias Baud
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A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes
MGJ Baud, E Lin-Shiao, T Cardote, C Tallant, A Pschibul, KH Chan, ...
Science 346 (6209), 638-641, 2014
Current strategies for the design of PROTAC linkers: a critical review
RI Troup, C Fallan, MGJ Baud
Exploration of Targeted Anti-tumor Therapy 1 (5), 273, 2020
Defining the mechanism of action and enzymatic selectivity of psammaplin A against its epigenetic targets
MGJ Baud, T Leiser, P Haus, S Samlal, AC Wong, RJ Wood, V Petrucci, ...
Journal of medicinal chemistry 55 (4), 1731-1750, 2012
Toward photopharmacological antimicrobial chemotherapy using photoswitchable amidohydrolase inhibitors
CE Weston, A Krämer, F Colin, O Yildiz, MGJ Baud, FJ Meyer-Almes, ...
ACS infectious diseases 3 (2), 152-161, 2017
Is NMR fragment screening fine-tuned to assess druggability of protein–protein interactions?
DM Dias, I Van Molle, MGJ Baud, C Galdeano, CFGC Geraldes, A Ciulli
ACS medicinal chemistry letters 5 (1), 23-28, 2014
Harnessing Fluorine–Sulfur Contacts and Multipolar Interactions for the Design of p53 Mutant Y220C Rescue Drugs
MR Bauer, RN Jones, MGJ Baud, R Wilcken, FM Boeckler, AR Fersht, ...
ACS chemical biology 11 (8), 2265-2274, 2016
Dual wavelength asymmetric photochemical synthesis with circularly polarized light
RD Richardson, MGJ Baud, CE Weston, HS Rzepa, MK Kuimova, ...
Chemical Science 6 (7), 3853-3862, 2015
Aminobenzothiazole derivatives stabilize the thermolabile p53 cancer mutant Y220C and show anticancer activity in p53-Y220C cell lines
MGJ Baud, MR Bauer, L Verduci, FA Dingler, KJ Patel, DH Roy, ...
European journal of medicinal chemistry 152, 101-114, 2018
New synthetic routes to triazolo-benzodiazepine analogues: expanding the scope of the bump-and-hole approach for selective bromo and extra-terminal (BET) bromodomain inhibition
MGJ Baud, E Lin-Shiao, M Zengerle, C Tallant, A Ciulli
Journal of medicinal chemistry 59 (4), 1492-1500, 2016
Exploiting Transient Protein States for the Design of Small-Molecule Stabilizers of Mutant p53
AC Joerger, MR Bauer, R Wilcken, MGJ Baud, H Harbrecht, TE Exner, ...
Structure 23 (12), 2246-2255, 2015
Optimization of a “bump-and-hole” approach to allele-selective BET bromodomain inhibition
AC Runcie, M Zengerle, KH Chan, A Testa, L van Beurden, MGJ Baud, ...
Chemical Science 9 (9), 2452-2468, 2018
Luminescent Lanthanide Helicates Self-Assembled from Ditopic Ligands Bearing Phosphonic Acid or Phosphoester Units
AS Chauvin, S Comby, M Baud, C De Piano, C Duhot, JCG Bünzli
Inorganic chemistry 48 (22), 10687-10696, 2009
Key Players in the Mutant p53 Team: Small Molecules, Gene Editing, Immunotherapy
V Chasov, R Mirgayazova, E Zmievskaya, R Khadiullina, A Valiullina, ...
Frontiers in Oncology 10, 2020
Thioester derivatives of the natural product psammaplin A as potent histone deacetylase inhibitors
MGJ Baud, T Leiser, V Petrucci, M Gunaratnam, S Neidle, ...
Beilstein journal of organic chemistry 9 (1), 81-88, 2013
New synthetic strategies towards psammaplin A, access to natural product analogues for biological evaluation
MGJ Baud, T Leiser, FJ Meyer-Almes, MJ Fuchter
Organic & Biomolecular Chemistry 9 (3), 659-662, 2011
Horil Roy, D.; Joerger, AC; Fersht, AR Aminobenzothiazole derivatives stabilize the thermolabile p53 cancer mutant Y220C and show anticancer activity in p53-Y220C cell lines
MGJ Baud, MR Bauer, L Verduci, FA Dingler, KJ Patel
Eur. J. Med. Chem 152, 101-114, 2018
Discovery of Nanomolar-Affinity Pharmacological Chaperones Stabilizing the Oncogenic p53 Mutant Y220C
JR Stephenson Clarke, LR Douglas, PJ Duriez, DI Balourdas, AC Joerger, ...
ACS Pharmacology & Translational Science 5 (11), 1169-1180, 2022
Kinetic method for the large-scale analysis of the binding mechanism of histone deacetylase inhibitors
C Meyners, MGJ Baud, MJ Fuchter, FJ Meyer-Almes
Analytical biochemistry 460, 39-46, 2014
Highly Ligand Efficient and Selective N‐2‐(Thioethyl) picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A
MGJ Baud, P Haus, T Leiser, FJ Meyer‐Almes, MJ Fuchter
ChemMedChem 8 (1), 149-156, 2013
Biophysical Survey of Small-Molecule β-Catenin Inhibitors: A Cautionary Tale
MA McCoy, D Spicer, N Wells, K Hoogewijs, M Fiedler, MGJ Baud
Journal of medicinal chemistry 65 (10), 7246-7261, 2022
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