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Violetta Cecchetti
Violetta Cecchetti
Full Professor in Medicinal Chemistry, Università di Perugia
Verified email at unipg.it - Homepage
Title
Cited by
Cited by
Year
A 1, 8-naphthyridone derivative targets the HIV-1 Tat-mediated transcription and potently inhibits the HIV-1 replication
S Massari, D Daelemans, ML Barreca, A Knezevich, S Sabatini, ...
Journal of medicinal chemistry 53 (2), 641-648, 2010
1572010
6-Aminoquinolones as new potential anti-HIV agents
V Cecchetti, C Parolin, S Moro, T Pecere, E Filipponi, A Calistri, ...
Journal of medicinal chemistry 43 (20), 3799-3802, 2000
1472000
Effects of novel 6-desfluoroquinolones and classic quinolones on pentylenetetrazole-induced seizures in mice
A De Sarro, V Cecchetti, V Fravolini, F Naccari, O Tabarrini, G De Sarro
Antimicrobial agents and chemotherapy 43 (7), 1729-1736, 1999
1471999
Evolution from a Natural Flavones Nucleus to Obtain 2-(4-Propoxyphenyl)quinoline Derivatives As Potent Inhibitors of the S. aureus NorA Efflux Pump
S Sabatini, F Gosetto, G Manfroni, O Tabarrini, GW Kaatz, D Patel, ...
Journal of medicinal chemistry 54 (16), 5722-5736, 2011
1212011
Quinolonecarboxylic acids. 2. Synthesis and antibacterial evaluation of 7-oxo-2, 3 dihydro-7H-pyrido [1, 2, 3-de][1, 4] benzothiazine-6-carboxylic acids
V Cecchetti, A Fravolini, R Fringuelli, G Mascellani, P Pagella, M Palmioli, ...
Journal of medicinal chemistry 30 (3), 465-473, 1987
1161987
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors
S Sabatini, F Gosetto, S Serritella, G Manfroni, O Tabarrini, N Iraci, ...
Journal of Medicinal Chemistry 55 (7), 3568-3572, 2012
992012
Synthesis and anti-BVDV activity of acridones as new potential antiviral agents
O Tabarrini, G Manfroni, A Fravolini, V Cecchetti, S Sabatini, E De Clercq, ...
Journal of medicinal chemistry 49 (8), 2621-2627, 2006
992006
A broad anti-influenza hybrid small molecule that potently disrupts the interaction of polymerase acidic protein–basic protein 1 (PA-PB1) subunits
S Massari, G Nannetti, J Desantis, G Muratore, S Sabatini, G Manfroni, ...
Journal of Medicinal Chemistry 58 (9), 3830-3842, 2015
982015
Studies on 6-aminoquinolones: synthesis and antibacterial evaluation of 6-amino-8-methylquinolones
V Cecchetti, A Fravolini, MC Lorenzini, O Tabarrini, P Terni, T Xin
Journal of medicinal chemistry 39 (2), 436-445, 1996
951996
Velnacrine thiaanalogues as potential agents for treating alzheimer's disease
O Tabarrini, V Cecchetti, A Temperini, E Filipponi, MG Lamperti, ...
Bioorganic & medicinal chemistry 9 (11), 2921-2928, 2001
932001
Structure− activity relationship study on anti-HIV 6-desfluoroquinolones
O Tabarrini, S Massari, D Daelemans, M Stevens, G Manfroni, S Sabatini, ...
Journal of medicinal chemistry 51 (17), 5454-5458, 2008
872008
New anti-human immunodeficiency virus type 1 6-aminoquinolones: mechanism of action
C Parolin, B Gatto, C Del Vecchio, T Pecere, E Tramontano, V Cecchetti, ...
Antimicrobial agents and chemotherapy 47 (3), 889-896, 2003
872003
Mg2+-mediated binding of 6-Substituted quinolones to DNA: Relevance to biological activity
C Sissi, M Andreolli, V Cecchetti, A Fravolini, B Gatto, M Palumbo
Bioorganic & medicinal chemistry 6 (9), 1555-1561, 1998
801998
Design and synthesis of modified quinolones as antitumoral acridones
O Tabarrini, V Cecchetti, A Fravolini, G Nocentini, A Barzi, S Sabatini, ...
Journal of medicinal chemistry 42 (12), 2136-2144, 1999
781999
Highly Potent 1,4-Benzothiazine Derivatives as KATP-Channel Openers
V Cecchetti, V Calderone, O Tabarrini, S Sabatini, E Filipponi, L Testai, ...
Journal of medicinal chemistry 46 (17), 3670-3679, 2003
692003
6-Aminoquinolones: a new class of quinolone antibacterials?
V Cecchetti, S Clementi, G Cruciani, A Fravolini, PG Pagella, A Savino, ...
Journal of medicinal chemistry 38 (6), 973-982, 1995
681995
Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors
A Astolfi, T Felicetti, N Iraci, G Manfroni, S Massari, D Pietrella, O Tabarrini, ...
Journal of medicinal chemistry 60 (4), 1598-1604, 2017
652017
Potent 6-desfluoro-8-methylquinolones as new lead compounds in antibacterial chemotherapy
V Cecchetti, A Fravolini, M Palumbo, C Sissi, O Tabarrini, P Terni, T Xin
Journal of medicinal chemistry 39 (25), 4952-4957, 1996
651996
Inhibition of subgenomic hepatitis C virus RNA replication by acridone derivatives: identification of an NS3 helicase inhibitor
G Manfroni, J Paeshuyse, S Massari, S Zanoli, B Gatto, G Maga, ...
Journal of medicinal chemistry 52 (10), 3354-3365, 2009
642009
Studies on anti-HIV quinolones: new insights on the C-6 position
S Massari, D Daelemans, G Manfroni, S Sabatini, O Tabarrini, ...
Bioorganic & medicinal chemistry 17 (2), 667-674, 2009
632009
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