| The first one-pot ambient-temperature synthesis of 1, 2, 4-oxadiazoles from amidoximes and carboxylic acid esters S Baykov, T Sharonova, A Shetnev, S Rozhkov, S Kalinin, AV Smirnov Tetrahedron 73 (7), 945-951, 2017 | 89 | 2017 |
| Continued exploration of 1, 2, 4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX … M Krasavin, A Shetnev, T Sharonova, S Baykov, S Kalinin, A Nocentini, ... European Journal of Medicinal Chemistry 164, 92-105, 2019 | 78 | 2019 |
| Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1, 2, 4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and … M Krasavin, A Shetnev, T Sharonova, S Baykov, T Tuccinardi, S Kalinin, ... Bioorganic Chemistry 76, 88-97, 2018 | 61 | 2018 |
| 1, 2, 4-oxadiazole/2-imidazoline hybrids: multi-target-directed compounds for the treatment of infectious diseases and cancer A Shetnev, S Baykov, S Kalinin, A Belova, V Sharoyko, A Rozhkov, ... International Journal of Molecular Sciences 20 (7), 1699, 2019 | 50 | 2019 |
| New tetracyclic 1, 4-oxazepines constructed via practically simple tandem condensation strategy from readily available synthons AV Sapegin, SA Kalinin, AV Smirnov, MV Dorogov, M Krasavin Tetrahedron 70 (5), 1077-1083, 2014 | 32 | 2014 |
| Carbonic anhydrase IX inhibitors as candidates for combination therapy of solid tumors S Kalinin, A Malkova, T Sharonova, V Sharoyko, A Bunev, CT Supuran, ... International Journal of Molecular Sciences 22 (24), 13405, 2021 | 31 | 2021 |
| Inhibitory activity against carbonic anhydrase IX and XII as a candidate selection criterion in the development of new anticancer agents M Krasavin, S Kalinin, T Sharonova, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 1555-1561, 2020 | 29 | 2020 |
| Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer … M Krasavin, A Shetnev, S Baykov, S Kalinin, A Nocentini, V Sharoyko, ... European Journal of Medicinal Chemistry 168, 301-314, 2019 | 28 | 2019 |
| Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases CT Supuran, S Kalinin, M Tanç, P Sarnpitak, P Mujumdar, SA Poulsen, ... Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup1), 197-202, 2016 | 28 | 2016 |
| Human carbonic anhydrase inhibitory profile of mono-and bis-sulfonamides synthesized via a direct sulfochlorination of 3-and 4-(hetero) arylisoxazol-5-amine scaffolds M Krasavin, M Korsakov, Z Zvonaryova, E Semyonychev, T Tuccinardi, ... Bioorganic & medicinal chemistry 25 (6), 1914-1925, 2017 | 25 | 2017 |
| Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1, 4] oxazepine-based carbonic anhydrase inhibitors A Sapegin, S Kalinin, A Angeli, CT Supuran, M Krasavin Bioorganic Chemistry 76, 140-146, 2018 | 24 | 2018 |
| Combining carbonic anhydrase and thioredoxin reductase inhibitory motifs within a single molecule dramatically increases its cytotoxicity M Krasavin, T Sharonova, V Sharoyko, D Zhukovsky, S Kalinin, ... Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 665-671, 2020 | 23 | 2020 |
| Mucoadhesive properties of nanogels based on stimuli-sensitive glycosaminoglycan-graft-pNIPAAm copolymers I Pilipenko, V Korzhikov-Vlakh, A Valtari, Y Anufrikov, S Kalinin, ... International Journal of Biological Macromolecules 186, 864-872, 2021 | 22 | 2021 |
| Primary mono-and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases M Krasavin, M Korsakov, O Ronzhina, T Tuccinardi, S Kalinin, M Tanç, ... Journal of Enzyme Inhibition and Medicinal Chemistry 32 (1), 920-934, 2017 | 22 | 2017 |
| Dibenzo [b, f] pyrazolo [1, 5-d][1, 4] oxazepines: Facile Construction of a Rare Heterocyclic System via Tandem Aromatic Nucleophilic Substitution–Smiles Rearrangement … AV Sapegin, SA Kalinin, AV Smirnov, MV Dorogov, M Krasavin Synthesis 44 (15), 2401-2407, 2012 | 21 | 2012 |
| Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo … D Dar'in, G Kantin, S Kalinin, T Sharonova, A Bunev, GI Ostapenko, ... European Journal of Medicinal Chemistry 222, 113589, 2021 | 19 | 2021 |
| Multicomponent chemistry in the synthesis of carbonic anhydrase inhibitors S Kalinin, CT Supuran, M Krasavin Journal of enzyme inhibition and medicinal chemistry 31 (sup4), 185-199, 2016 | 19 | 2016 |
| Highly hydrophilic 1, 3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure S Kalinin, A Valtari, M Ruponen, E Toropainen, A Kovalenko, A Nocentini, ... Bioorganic & Medicinal Chemistry 27 (21), 115086, 2019 | 15 | 2019 |
| Radiotracers for positron emission tomography (PET) targeting tumour-associated carbonic anhydrase isoforms V Burianova, S Kalinin, CT Supuran, M Krasavin European Journal of Medicinal Chemistry 213, 113046, 2021 | 14 | 2021 |
| From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction S Kalinin, A Nocentini, A Kovalenko, V Sharoyko, A Bonardi, A Angeli, ... European Journal of Medicinal Chemistry 182, 111642, 2019 | 14 | 2019 |
