Bradyzide, a potent non‐peptide B2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia GM Burgess, MN Perkins, HP Rang, EA Campbell, MC Brown, P McIntyre, ... British journal of pharmacology 129 (1), 77-86, 2000 | 126 | 2000 |
Cloned murine bradykinin receptor exhibits a mixed B1 and B2 pharmacological selectivity. P McIntyre, E Phillips, E Skidmore, M Brown, M Webb Molecular pharmacology 44 (2), 346-355, 1993 | 92 | 1993 |
The design of non-peptide human bradykinin B 2 receptor antagonists employing the benzodiazepine peptidomimetic scaffold EK Dziadulewicz, MC Brown, AR Dunstan, W Lee, NB Said, PJ Garratt Bioorganic & medicinal chemistry letters 9 (3), 463-468, 1999 | 83 | 1999 |
2-Nitrophenylcarbamoyl-(S)-prolyl-(S)-3-(2-naphthyl) alanyl-N-benzyl-N-methylamide (SDZ NKT 343), a potent human NK1 tachykinin receptor antagonist with good oral analgesic … C Walpole, SY Ko, M Brown, D Beattie, E Campbell, F Dickenson, S Ewan, ... Journal of medicinal chemistry 41 (17), 3159-3173, 1998 | 83 | 1998 |
1-(2-Nitrophenyl) thiosemicarbazides: a novel class of potent, orally active non-peptide antagonist for the bradykinin B2 receptor EK Dziadulewicz, TJ Ritchie, A Hallett, CR Snell, SY Ko, R Wrigglesworth, ... Journal of medicinal chemistry 43 (5), 769-771, 2000 | 31 | 2000 |
Nonpeptide Bradykinin B2 Receptor Antagonists: Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B2 Receptor Antagonists 1 EK Dziadulewicz, TJ Ritchie, A Hallett, CR Snell, JW Davies, ... Journal of medicinal chemistry 45 (11), 2160-2172, 2002 | 29 | 2002 |
Comparative, general pharmacology of SDZ NKT 343, a novel, selective NK1 receptor antagonist CSJ Walpole, MCS Brown, IF James, EA Campbell, P McIntyre, ... British journal of pharmacology 124 (1), 83-92, 1998 | 23 | 1998 |
Interaction of amyloid β protein (25–35) with tachykinin receptors P Rovero, R Patacchini, AR Renzetti, M Brown, J Mizrahi, CA Maggi, ... Neuropeptides 22 (2), 99-101, 1992 | 21 | 1992 |
Actinomycin D is a competitive and selective antagonist at NK2 tachykinin receptors R Patacchini, M Astolfi, MCS Brown, CA Maggi Neuropeptides 20 (2), 109-114, 1991 | 14 | 1991 |
Selective labelling of bradykinin receptor subtypes in WI38 human lung fibroblasts SB Phagoo, M Yaqoob, M Brown, GM Burgess British journal of pharmacology 119 (5), 863-868, 1996 | 13 | 1996 |
Molecular studies on kinin receptors M Brown, M Webb, E Phillips, E Skidmore, P McIntyre Canadian journal of physiology and pharmacology 73 (7), 780-786, 1995 | 9 | 1995 |
[125I] His-neurokinin A binds selectively to NK2 receptors of the B-type in rat small intestine smooth muscle membranes MCS Brown, M Biagi, AR Renzetti, P Rovero, M Criscuoli, J Mizrahi European Journal of Pharmacology: Molecular Pharmacology 227 (2), 163-171, 1992 | 9 | 1992 |
Further characterisation of the [35S]-TBPS binding site of the GABA receptor complex in locust (Schistocerca gregaria) ganglia membranes MCS Brown, GC Lunt, A Stapleton Comparative Biochemistry and Physiology Part C: Comparative Pharmacology 92 …, 1989 | 9 | 1989 |
The biochemical characterization of insect GABA receptors GG Lunt, MCS Brown, K Riley, DM Rutherford Neurotox 88, 185-192, 1988 | 8 | 1988 |
t-Butylbicyclophosphoro [35S] thionate binding to ganglionic membranes of the locust (Schistocerca gregaria) MCS BROWN, GG LUNT, A STAPLETON Biochemical Society Transactions 15 (3), 503-504, 1987 | 2 | 1987 |
Human Neurokinin-1 receptors, transiently transfected into Cos-7 cells, couple to simian G-proteins SG EWAN, CL SEAR, E SKIDMORE, P McINTYRE, MCS BROWN Biochemical Society Transactions 23 (1), 95S-95S, 1995 | | 1995 |
Cloned Murine Bradykinin Receptor Exhibits a Mixed B1 and B2 Pharmacological Selectivity P McIntyre, E Phillips, E Skidmore, M Brown, M Webb Molecular Pharmacology 45 (3), 561, 1994 | | 1994 |
A single cloned mouse bradykinin (Bk) receptor exhibits the pharmacology of both B 1 and B 2 receptors M Brown, M Webb, E Phillips, E Skidmore, P McIntyre Neuropeptides 24 (4), 241-242, 1993 | | 1993 |
Calcitonin gene-related peptide (CGRP) interacts with NK2B receptors in rat small intestine smooth muscle membranes MCS Brown, M Biagi, AR Renzetti, J Mizrahi Neuropeptides 22 (1), 11, 1992 | | 1992 |
Effects of GTP analogues on neurokinins receptor subtypes AR Renzetti, MCS Brown, J Mizrahi Neuropeptides 22 (1), 56, 1992 | | 1992 |